For research purposes only

Cat. No BA94673154

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Description of biological activity

group II metabotropic glutamate receptor (mGluR) antagonist

TECHNICAL INFORMATION

(-)-(1R,2R,3R,5R,6R)-2-amino-3-(3,4-dichlorobenzyloxy)-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic acid (MGS0039) group II metabotropic glutamate receptor (mGluR) antagonist

IUPAC Name: (-)-(1R,2R,3R,5R,6R)-2-amino-3-(3,4-dichlorobenzyloxy)-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic acid (MGS0039)

CAS Number: 569686-87-9

Purity: > 96% chemical purity (LCMS)

1H-NMR spectrum (click to enlarge)

REFERENCES

1. Bioorg. Med. Chem. 2006,В 12, 4193-4207, 2. J. Med. Chem. 2004, 47, 4570-4587

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