For research purposes only

Cat. No BA94673157

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Description of biological activity

Inhibition of trace amine associated receptor 1 (TTAR1). In a radioligand assay on HEK293 cells stably transfected with pIRESneo2 expression plasmids containing mouse trace amine associated receptor 1 (TAAR1) coding sequences the compound showed Ki = 1 nM [US2009/36420 A1, 2009].

TECHNICAL INFORMATION

N-(3-ethoxy-phenyl)-4-pyrrolidin-1-yl-3-trifluoromethyl-benzamide inhibition of trace amine associated receptor 1 (TTAR1).

IUPAC Name: N-(3-ethoxy-phenyl)-4-pyrrolidin-1-yl-3-trifluoromethyl-benzamide

CAS Number: 1110781-88-8

Purity: > 96% chemical purity (LCMS)

1H-NMR spectrum (click to enlarge)

REFERENCES

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