For research purposes only

Cat. No BA131318434

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Description of biological activity

Reversible competitive inhibitor of Porcine Pancreatic Elastase (PPE) and Human Leukocyte Elastase (HLE) For the Porcine Pancreatic Elastase Ki = 0.22 mM and for Human Leukocyte Elastase Ki = 2 mM.

Keywords:

TECHNICAL INFORMATION

1-[6-Amino-2-(2,2,2-trifluoro-acetylamino)-hexanoyl]-pyrrolidine-2-carboxylic acid (4-isopropyl-phenyl)-amide inhibitor of PPE and HLE

IUPAC Name: 1-[6-Amino-2-(2,2,2-trifluoro-acetylamino)-hexanoyl]-pyrrolidine-2-carboxylic acid (4-isopropyl-phenyl)-amide

CAS Number: 86800-68-2

Purity: > 96% chemical purity (LCMS)
> 95 de

REFERENCES

1. J.Biol.Chem.,1983, 258, 8312
2. Biochem. 1995, 34, 3193

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